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Palbociclib (PD0332991) Isethionate
CAS No. 827022-33-3
Palbociclib (PD0332991) Isethionate ( —— )
Catalog No. M16070 CAS No. 827022-33-3
Palbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 with IC50 of 11 nM/16 nM.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 42 | In Stock |
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| 10MG | 60 | In Stock |
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| 50MG | 78 | In Stock |
|
| 100MG | 114 | In Stock |
|
| 200MG | 141 | In Stock |
|
| 500MG | 294 | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePalbociclib (PD0332991) Isethionate
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NoteResearch use only, not for human use.
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Brief DescriptionPalbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 with IC50 of 11 nM/16 nM.
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DescriptionPalbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 with IC50 of 11 nM/16 nM. It shows no activity against CDK1/2/5, EGFR, FGFR, PDGFR, InsR, etc. Phase 3.
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Synonyms——
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PathwayAngiogenesis
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TargetCDK
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RecptorCDK2/CyclinA; CDK2/CyclinE2; CDK4/CyclinD1; CDK4/CyclinD3; CDK6/CyclinD2
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number827022-33-3
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Formula Weight573.66
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Molecular FormulaC24H29N7O2·C2H6O4S
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Purity>98%(HPLC)
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SolubilityWater: 50 mg/mL warmed (87.15 mM)
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SMILESOCCS(O)(=O)=O.CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(C=C3)N3CCNCC3)N=C2N(C2CCCC2)C1=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Fry DW, et al. Mol Y Ther, 2004, 3(11), 1427-1438.
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